Tamibarotene - CAS# 94497-51-5 oxifen citrate inhibition of TPH1 occurred in

inhibition of TPH1 occurred in 10(-8) -10(-7) mol L(-1) range

Formula: C22H22N6O3

Leuprolide acetate is the acetate salt of a synthetic nonapeptide analogue of gonadotropin-releasing hormone

5-c]pyridine-6-carboxylic acid

InChiKey: ACGUYXCXAPNIKK-UHFFFAOYSA-N

Tamibarotene - CAS# 94497-51-5 oxifen citrate inhibition of TPH1 occurred inTamibarotene, also known as SY 1425, is an orally active, synthetic retinoid, developed to overcome all trans retinoic acid (ATRA) resistance, with potential antineoplastic activity. As a specific retinoic acid receptor (RAR) alpha beta agonist, tamibarotene is approximately ten times more potent than ATRA in inducing cell differentiation and apoptosis in HL 60 (human promyelocytic leukemia) cell lines in vitro. Due to a lower affinity for cellular